TY - BOOK AU - Kar, Ashutosh TI - Medicinal chemistry: introduction - classification - synthesis - explanation - mechanism of action - structure activity relationships (SARs) - usages - doses SN - 9788122430868 AV - RS403.K37 PY - 2010/// CY - New Delhi PB - New Age Techno Press N1 - Includes index; Content: Drug design - A rational approach -- Physical-chemical factors and biological activities -- Molecular modelling and design -- General anaesthetics -- Local anaesthetics -- Sedatives and hypnotics -- Anticonvulsants -- Muscle relaxants -- Central nervous system stimulants -- Antipyretic analgesics -- Narcotic analgesics (opiate analgesics) -- Cardiovascular drugs -- Autonomic drugs -- Diuretics -- Antihistamincs -- Non-steroidal anti-inflammatory drugs (NSAIDs) -- Antiparkinsonism agents -- Expectorants and antitussives -- Sulphonamides -- Antimalarials -- Anthelmintics -- Insulin and oral hypoglycemic agents -- Steroids -- Adrenocortal steroids -- Antibiotics -- Antimycobacterial drugs -- Antineoplastic agents -- Antipsychotics (tranquilizers) -- Antiviral drugs -- Newer drugs for newer diseases -- Pro-drug approach in drug design -- Drug discovery via enzyme inhibition. ER -